Development of a monoclonal anti-ADAMTS-5 antibody that specifically blocks the interaction with LRP1

نویسندگان

  • Salvatore Santamaria
  • Oleg Fedorov
  • John McCafferty
  • Gillian Murphy
  • Jayesh Dudhia
  • Hideaki Nagase
  • Kazuhiro Yamamoto
چکیده

The potent aggrecanase ADAMTS-5 is constitutively secreted by chondrocytes, but it is rapidly endocytosed in normal cartilage via the cell surface endocytic receptor LRP1. Therefore it is difficult to detect the total ADAMTS-5 activity produced. In this study, we isolated a monoclonal anti-ADAMTS-5 antibody 1B7 that blocks LRP1-mediated internalization without affecting the aggrecanolytic activity. Addition of 1B7 to cultured human chondrocytes revealed the full aggrecanolytic activity of ADAMTS-5 generated by the cells. 1B7 is a useful tool to estimate the ADAMTS-5 activity and to identify its potential roles in the tissues.

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عنوان ژورنال:

دوره 9  شماره 

صفحات  -

تاریخ انتشار 2017